| S.No. | API Intermediate | CAS NO |
|---|---|---|
| Intermediate Name | ||
| 1. | 2-(7-Methoxy-1-naphthyl)ethylamine hydrochloride | 139525-77-2 |
| 2. | 7-Methoxy-1-naphthylacetonitrile | 138113-08-3 |
| 3. | 2-(7-Methoxy-1-naphthyl)ethylamine | 138113-09-4 |
| 4. | Ethyl (7-methoxy-1,2,3,4-tetrahydro-1-naphthylidene)acetate | – |
| Aprepitant | ||
| 5. | (2R)-4-Benzyl-2-{(1R)-1-[3,5-Bis(trifluoromethyl) phenyl]ethoxy}morpholin-3-one | 287930-75-0 |
| 6. | 1-[3,5-bis(trifluoromethyl)phenyl]ethylbromide | 160376-84-1 |
| 7. | (2R,3S)-2-[(1R)-1-[3,5-bis(trifluoromethyl) phenyl]ethoxy]-3-(4-fluorophenyl)-Morpholine | 171482-05-6 |
| 8. | Ethyl (7-methoxy-1,2,3,4-tetrahydro-1-naphthylidene)acetate | – |
| Dabigartan | ||
| 9. | {[4-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)phenyl]amino}acetic acid | 872728-82-0 |
| 10. | Ethyl 3-[{[3-methyl-4-(methylamino)phenyl]carbonyl}(pyridin-2-yl)amino]propanoate | 212332-56-0 |
| Infigratinib | ||
| 11. | 5-Amino-3 (trifluoromethyl) pyridine-2-carbonitrile | 573762-62-6 |
| 12. | 1-(6-Chloropyrimidin-4-yl)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-methyl urea | – |
| Darifenacin | ||
| 13. | 1-Tosyl-3-(R)-(-)-hydroxy pyrrolidine | 133034-00-1 |
| 14. | 5-Chloroethyl-2,3- dihydrobenzofuran | 943034-50-2 |
| 15. | 3-(S)-(1-cyano-1,1-diphenylmethyl)-1-[2-(2,3-dihydrobenzofuran-5-yl)ethyl] pyrrolidine hydrobromide | – |
| Desloratadine | ||
| 16. | 8-chloro-11-piperidin-4-ylidene-6,11-dihydro-5H-benzo[5,6]cyclohepta [1,2-b]pyridine | 100643-71-8 |
| 17. | 8-Bromo-6,11-dihydro-11-(1-methyl-4-piperdinylidene)-5H-benzo[5,6] cyclohepta [1,2-b]pyridine | 130642-57-8 |
| Dutasteride | ||
| 18. | 3- Oxo-4-aza-5α-androst-1-ene 17β-carboxamide | 104239-97-6 |
| Ezetimibe | ||
| 19. | (3R,4S)-1-(4-fluorophenyl)-3-[(3S)-3-(4-fluorophenyl)-3-hydroxypropyl]-4- (4-benzyloxyphenyl)azetidin-2-one | 163222-32-0 |
| Finasteride | ||
| 20. | 3-oxo-4-aza-5 alpha-androstan-17 beta-carboxylic acid | 103335-55-3 |
| 21. | 17β-(N-tert-Butylcarbamoyl-)3-Oxo-4-aza-5α-androstane | 98319-24-5 |
| Mirogabalin | ||
| 22. | [1R, 5S-]-3-Ethyl bicycle[3,2,0]hept-3-ene-6-one | – |
| Lamotrigine | ||
| 23. | 6-(2,3-Dichlorophenyl)-1,2,4-triazine-3,5-diamine | 84057-84-1 |
| Lenalidomide | ||
| 24. | 3 Amino-piperidine-2,6-dione hydrochloride | 24666-56-6 |
| 25. | 2-Bromomethyl-3-nitrobenzoic acid methyl ester | 98475-07-1 |
| 26. | 3-(4-Nitro-1-oxo-1, 3-dihydro-isoindol-2yl)-piperidine-2,6-dione | 827026-45-9 |
| Paliperidone | ||
| 27. | 3-(2-Chloroethyl)-6,7,8,9 Tetra Hydro-9 Hydroxy-2-Methyl-4H Pyrrido- (1,2-Alpha)-Pyrimidine-4-One | 130049-82-0 |
| 28. | 6-Fluoro-3-(4-Piperidinyl)1,2-Benzisoxazole Hydrochloride | 84163-13-3 |
| Palonosetron | ||
| 29. | (S)-N-(1-Azabicyclo[2.2.2]oct-3-yl)-5,6,7,8-tetrahydro-1-naphthalene carboxamide | 135729-78-1 |
| 30. | 5,6,7,8-Tetrahydronaphthoic acid | 4242-18-6 |
| Risperidone | ||
| 31. | 6-Fluoro-3-(4-Piperidinyl)-1,2-Benzisoxazole Hydrochloride | 84163-13-3 |
| 32. | 3-(2-Chloroethyl)-2-Methyl-6,7,8,9-Tetrahydro-4H-Pyrido-(1,2-a) Pyridine -4-one hydrochloride | 93076-03-0 |
| Rivaroxaban | ||
| 33. | 4-(4-Aminophenyl)morpholin-3-one | 438056-69-0 |
| 34. | 5-Chlorothiophene-2-carboxylic Acid | 24065-33-6 |
| 35. | (R)-4-[4-[(3-Chloro-2-hydroxypropyl)amino]phenyl]morpholin-3-one | – |
| Rivastigmine | ||
| 36. | (S)-1-(3-Methoxyphenyl)ethylamine | 82796-69-8 |
| 37. | S-(-)-[1-(3-methoxyphenyl)ethyl]-N,N-dimethylamine | 889443-69-0 |
| 38. | (S)-3-[1-(Dimethylamino)ethyl]phenol | 139306-10-8 |
| Rocuronium Bromide | ||
| 39. | (2b,3a,5a,16b,17b)-2-(4-Morpholinyl)-16-(1-pyrrolidinyl)androstane-3,17-diol | 119302-20-4 |
| 40. | (2b,3a,5a,16b,17b)-17-Acetoxy-3-hydroxy-2-(4-morpholinyl)-16-(1-pyrrolidinyl)androstane | 119302-24-8 |
| 41. | 2a 3a 16a 17a-diepoxy-17b-acetoxy-5a-androstane | 50588-22-2 |
| 42. | (2a,3a,5a,16b,17b)-2,3-Epoxy-16-(1-pyrrolidinyl)androstan-17-ol | 119302-19-1 |
| Sitagliptin Phosphate Monohydrate | ||
| 43. | 4-Oxo-4-[3-trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a] pyrazin-7(8H)-yl]- 1-(2,4,5-trifluorophenyl)butan-2-one | 119302-20-4 |
| 44. | (2Z)-4-Oxo-4-[3-trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a] pyrazin-7(8H)-yl] -1-(2,4,5-trifluorophenyl)butan-2-en-2-amine | 119302-24-8 |
| 45. | 3-Amino-1-[3-trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a] pyrazin-7(8H)-yl] -4-(2,4,5-trifluorophenyl)-1-butanone | 50588-22-2 |
| 46. | 3-(Trifluoromethyl)-5,6,7,8-tetrahydro [1,2,4]triazolo [4,3-a] pyrazine Hydrochloride | 119302-19-1 |
| Solifenacin | ||
| 47. | 1-Phenyl-1,2,3,4-tetrahydro-isoquinoline | 22990-19-8 |
| 48. | (1S)-1-Phenyl-1,2,3,4-tetrahydroisoquinoline | 118864-75-8 |
| Teneligliptin | ||
| 49. | 1-(5-methyl-2-phenylpyrazol-3-yl)piperazine | 401566-79-8 |
| 50. | (S)-tert-butyl 3-oxo-2-(thiazolidine-3-carbonyl)pyrrolidine-1-carboxylate | 401564-36-1 |
| Tolterodine Tartrate | ||
| 51. | 6-Methyl-4-phenylchroman-2-one | 40546-94-9 |
| 52. | Methyl 3-(2-methoxy-5-methylphenyl)-3-phenylpropanoate | 401564-36-1 |
| Valacyclovir | ||
| 53. | N-[(Phenylmethoxy)carbonyl]-L-valine 2-[(2-amino-1,6-dihydro-6-oxo- 9H-purin-9-yl)methoxy]ethyl ester | 124832-31-1 |
| Zafirlukast | ||
| 54. | Methyl 4-(bromomethyl)-3-methoxybenzoate | 70264-94-7 |
| 55. | {3 -[2-methoxy-4-carboxy-benZyl]-1 methyl-1H-indol-5-yl}-carbamic acid cyclopentyl ester | – |
| Zolmitriptan | ||
| 56. | (4S)-4-[(4-Aminophenyl)methyl]-2-oxazolidinone | 152305-23-2 |
| 57. | ethyl/methyl-3-[2-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)ethyl]-5-[(4S)-2-oxo- 1,3-oxazolan-4yl methyl]-1H-2-indole carboxylate | – |
| Zonisamide | ||
| 58. | 1,2-Benzisoxazole-3-acetic acid | 4865-84-3 |
| 59. | 1,2-Benzisoxazole-3-methanesulfonamide | 68291-97-4 |
| Fluoxetine | ||
| 60. | (±)-N-Methyl-γ-[4-(trifluoromethyl)phenoxy] benzenepropanamine | 54910-89-3 |
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